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Search Results for " human a-cgrp "

14

Compounds

Cat No. Product Name Synonyms Targets
TP2044L α-CGRP (human) acetate α-CGRP (human) acetate (90954-53-3 free base) Others
α-CGRP (human) acetate is a regulatory neuropeptide of 37 amino acids. It is the most potent vasodilator known to date and has inotropic and chronotropic effects.
TP2044 α-CGRP(human) α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.
TP1134 HCGRP-(8-37) Human α-CGRP (8-37)
Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist
T36555 Tyr-α-CGRP (human) (trifluoroacetate salt)
Tyr-α-CGRP is an N-terminal extended tyrosinated analogue of α-calcitonin gene-related peptide . It binds to amylin receptors AMY1 and AMY3 in COS-7 cells expressing the human receptors (IC50s = 141 and 1.86 nM, respecti...
TP1134L HCGRP-(8-37) acetate HCGRP-(8-37) acetate (119911-68-1 free base) CGRP Receptor
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.
T76874 Erenumab AMG-334 CGRP Receptor
Erenumab is a whole-human monoclonal antibody. Erenumab inhibits calcitonin gene-related peptide (CGRP) receptors. Erenumab can be used to prevent migraine attacks.
TP1130 β-CGRP, human CGRP-II (Human),Human β-CGRP
β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular and nervous systems. β-CGRP contains a disulphide bridge at th...
T75978 β-CGRP, human TFA
Human β-CGRP TFA (β-CGRP, human TFA) is a calcitonin peptide that functions through interaction with the calcitonin-receptor-like receptor (CRLR) and receptor-activity-modifying protein (RAMP) complex, demonstrating IC50...
T6590 MK-3207 Hydrochloride MK-3207 HCl CGRP Receptor
MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.
T75788 α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a potent vasodilator [1].
T12293 Olcegepant hydrochloride BIBN-4096 hydrochloride,BIBN4096BS hydrochloride Others
Olcegepant hydrochloride is a potent and selective non-peptidethe calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (with IC50 of 0.03 nM for human CGRP).
T76473 Adrenotensin (human)
Adrenotensin (human) (Pro-ADM-153-185 (human)), a 153-185 fragment of the Adrenomedullin precursor peptide, is part of the Multifunctional Adrenomedullin (ADM). This 52-amino acid peptide, a member of the CGRP superfamil...
T21558 MK-3207
MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC 50 = 0.12 nM; K i = 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. IC50 Value: 0.024 nM (Ki, Human CGRP) [1] As other CGRP recep...
T76678 Eptinezumab
Eptinezumab, a human monoclonal antibody, specifically binds to and blocks the calcitonin gene-related peptide (CGRP) from binding to its receptor, thus acting as a preventive treatment for migraine in adults [1].
TargetMol